David A Piotrowski

US Patent:

6479510, Nov 12, 2002

Filed:

Aug 17, 2001

Appl. No.:

09/932598

Inventors:

Jason K. Myers - Kalamazoo MI
David W. Piotrowski - Portage MI

Assignee:

Pharmacia Upjohn Company - Kalamazoo MI

International Classification:

A61K 31439

US Classification:

514305, 546133, 544127, 5142332

Abstract:

The invention provides compounds of Formula I: These compounds may be in the form of pharmaceutical salts or compositions, and racemic mixtures or pure enantiomers thereof. The compounds of Formula I are useful in pharmaceuticals in which 7 is known to be involved.

US Patent:

6486172, Nov 26, 2002

Filed:

Aug 17, 2001

Appl. No.:

09/932597

Inventors:

Jason K. Myers - Kalamazoo MI
David W. Piotrowski - Portage MI

Assignee:

Pharmacia Upjohn Company - Kalamazoo MI

International Classification:

A61K 31439

US Classification:

514305, 5142332, 546133, 544127

Abstract:

The invention provides compounds of Formula I: These compounds may be in the form of pharmaceutical salts or compositions, and racemic mixtures or pure enantiomers thereof. The compounds of Formula I are useful in pharmaceuticals in which 7 is known to be involved.

US Patent:

6492385, Dec 10, 2002

Filed:

Aug 17, 2001

Appl. No.:

09/932309

Inventors:

Jason K. Myers - Kalamazoo MI
Bruce N. Rogers - Portage MI
David W. Piotrowski - Portage MI
Alice L. Bodnar - Kalamazoo MI
Eric Jon Jacobsen - Richland MI
Jeffrey W. Corbett - Portage MI

Assignee:

Pharmacia Upjohn Company - Kalamazoo MI

International Classification:

A61K 31439

US Classification:

514305, 546133, 546135, 544127, 5142332

Abstract:

The invention provides compounds of Formula I: These compounds may be in the form of pharmaceutical salts or compositions, and racemic mixtures or pure enantiomers thereof. The compounds of Formula I are useful in pharmaceuticals in which 7 is known to be involved.

US Patent:

6492386, Dec 10, 2002

Filed:

Aug 17, 2001

Appl. No.:

09/932325

Inventors:

Jason K. Myers - Kalamazoo MI
David W. Piotrowski - Portage MI

Assignee:

Pharmacia Upjohn Company - Kalamazoo MI

International Classification:

A61K 31439

US Classification:

514305, 5142332, 546133, 544127

Abstract:

The invention provides compounds of Formula I: These compounds may be in the form of pharmaceutical salts or compositions, and racemic mixtures or pure enantiomers thereof. The compounds of Formula I are useful in pharmaceuticals in which 7 is known to be involved.

US Patent:

6500840, Dec 31, 2002

Filed:

Aug 17, 2001

Appl. No.:

09/932612

Inventors:

Jason K. Myers - Kalamazoo MI
Bruce N. Rogers - Portage MI
David W. Piotrowski - Portage MI
Alice L. Bodnar - Kalamazoo MI
Eric Jon Jacobsen - Richland MI
Jeffrey W. Corbett - Portage MI

Assignee:

Pharmacia Upjohn Company - Kalamazoo MI

International Classification:

A61K 31439

US Classification:

514305, 5142332, 546133, 546135, 544127

Abstract:

The invention provides compounds of Formula I: These compounds may be in the form of pharmaceutical salts or compositions, and racemic mixtures or pure enantiomers thereof. The compounds of Formula I are useful in pharmaceuticals in which 7 is known to be involved.

US Patent:

6562816, May 13, 2003

Filed:

Aug 14, 2002

Appl. No.:

10/218772

Inventors:

Donn G. Wishka - Kalamazoo MI
Jason K. Myers - Kalamazoo MI
Bruce N. Rogers - Portage MI
Eric Jon Jacobsen - Richland MI
David W. Piotrowski - Portage MI
Jeffrey W. Corbett - Portage MI
Alice L. Bodnar - Kalamazoo MI

Assignee:

Pharmacia Upjohn Company - Kalamazoo MI

International Classification:

A61K 315377

US Classification:

5142332, 514413, 544143, 546167, 546200, 5462697, 5462704, 5462714, 5462767, 548131, 548136, 548142, 548143, 548214, 548225, 548227, 548228, 548229, 548181, 548236, 548248, 5483121, 548453

Abstract:

The invention provides compounds of Formula I: compounds of the Formula I: wherein R , R , R , R , X, and W are defined herein. These compounds may be in the form of pharmaceutical salts or compositions, may be in pure enantiomeric form or racemic mixtures, and are useful in pharmaceuticals used to treat diseases or conditions in which 7 is known to be involved.

US Patent:

6599916, Jul 29, 2003

Filed:

Aug 17, 2001

Appl. No.:

09/932299

Inventors:

Jason K. Myers - Kalamazoo MI
Bruce N. Rogers - Portage MI
David W. Piotrowski - Portage MI
Alice L. Bodnar - Kalamazoo MI
Eric Jon Jacobsen - Richland MI
Jeffrey W. Corbett - Portage MI

Assignee:

Pharmacia Upjohn Company - Kalamazoo MI

International Classification:

A61K 31439

US Classification:

514305, 546133, 546135

Abstract:

The invention provides compounds of Formula I: These compounds may be in the form of pharmaceutical salts or compositions, and racemic mixtures or pure enantiomers thereof. The compounds of Formula I are useful in pharmaceuticals in which 7 is known to be involved.

US Patent:

6818641, Nov 16, 2004

Filed:

Aug 28, 2002

Appl. No.:

10/220446

Inventors:

David Walter Piotrowski - Portage MI

Assignee:

E. I. du Pont de Nemours and Company - Wilmington DE

International Classification:

C07D25306

US Classification:

514242, 514243, 544182, 544183, 544184

Abstract:

Compounds of Formula (I), and their N-oxides and agriculturally suitable salts, are disclosed which are useful as arthropodicides wherein A is H; E is H or C -C alkyl; or A and E can be taken together to form âCH â, âCH CH â, âOâ, âSâ, âS(O)â, âS(O) â, âNR â, âOCH â, âSCH â, âN(R )CH â, substituted âCH â and substituted âCH CH â, the substituents independently selected from 1-2 halogen and 1-2 methyl; W is N or CR ; X is CR R , O, S, NR or a direct bond, provided that when W is N, then X is other than a direct bond; Y is H, C -C alkyl, C -C alkenyl, C -C alkynyl, C -C alkylsulfonyl, C -C cycloalkyl, C -C cycloalkylalkyl, NR R , N CR R , OR , COR , CO R or C -C alkyl substituted by at least one group selected from halogen, C -C alkoxy, CN, NO , S(O) R , COR , CO R and optionally substituted phenyl; Z is O or S; and R , R , R , R , R , R , R , R , R , R , R , R , R , R , G, n and r are as defined in the disclosure. Also disclosed are compositions containing the compounds of Formula (I) and a method for controlling arthropods which involves contacting the arthropods or their environment with an effective amount of a compound of Formula (I).