Todd K. Jones - Solana Beach CA Mark E. Goldman - San Diego CA Charlotte L. F. Pooley - San Diego CA David T. Winn - San Diego CA James P. Edwards - San Diego CA Sarah J. West - San Diego CA Christopher M. Tegley - San Diego CA Lin Zhi - San Diego CA Lawrence G. Hamann - San Diego CA Luc J. Farmer - La Jolla CA Robert L. Davis - Santee CA
Non-steroidal compounds which are high affinity, high selectivity modulators for steroid receptors are disclosed. Also disclosed are pharmaceutical compositions incorporating such compounds, methods for employing the disclosed compounds and compositions for treating patients requiring steroid receptor agonist or antagonist therapy, intermediates useful in the preparation of the compounds and processes for the preparation of the steroid receptor modulator compounds.
Todd Jones - Solana Beach CA, US Mark Goldman - San Diego CA, US Charlotte Pooley - San Diego CA, US David Winn - San Diego CA, US James Edwards - San Diego CA, US Sarah West - San Diego CA, US Christopher Tegley - San Diego CA, US Lin Zhi - San Diego CA, US Lawrence Hamann - San Diego CA, US Luc Farmer - La Jolla CA, US Robert Davis - Santee CA, US
International Classification:
A61K031/47
US Classification:
514/312000, 514/314000
Abstract:
Non-steroidal compounds which are high affinity, high selectivity modulators for steroid receptors are disclosed. Also disclosed are pharmaceutical compositions incorporating such compounds, methods for employing the disclosed compounds and compositions for treating patients requiring steroid receptor agonist or antagonist therapy, intermediates useful in the preparation of the compounds and processes for the preparation of the steroid receptor modulator compounds.
Todd K. Jones - Solana Beach CA Lin Zhi - San Diego CA Christopher M. Tegley - San Diego CA David T. Winn - San Diego CA Lawrence G. Hamann - San Diego CA James P. Edwards - San Diego CA Sarah J. West - San Diego CA
Assignee:
Ligand Pharmaceuticals Incorporated - San Diego CA
International Classification:
A61K 3147 C07D47104 C07D22116 C07D49148 C07D49152
US Classification:
514285
Abstract:
Non-steroidal compounds which are high affinity, high selectivity modulators for steroid receptors are disclosed. Also disclosed are pharmaceutical compositions incorporating such compounds, methods for employing the disclosed compounds and compositions for treating patients requiring steroid receptor agonist or antagonist therapy, intermediates useful in the preparation of the compounds and processes for the preparation of the steroid receptor modulator compounds.
Tricyclic Steroid Receptor Modulator Compounds And Methods
Todd K. Jones - Solana Beach CA David T. Winn - San Diego CA Mark E. Goldman - San Diego CA Lawrence G. Hamann - San Diego CA Lin Zhi - San Diego CA Luc J. Farmer - La Jolla CA Robert L. Davis - Santee CA
Assignee:
Ligand Pharmaceuticals Incorporated - San Diego CA
International Classification:
A61K 3144 A61K 3147 A61K 3140 C07D47152 C07D47104
US Classification:
514291
Abstract:
Non-steroidal compounds which are high affinity, high selectivity modulators for steroid receptors are disclosed. Also disclosed are pharmaceutical compositions incorporating such compounds, methods for employing the disclosed compounds and compositions for treating patients requiring steroid receptor agonist or antagonist therapy, intermediates useful in the preparation of the compounds and processes for the preparation of the steroid receptor modulator compounds.
Todd K. Jones - Solana Beach CA Mark E. Goldman - San Diego CA Charlotte L.F. Pooley - San Diego CA David T. Winn - San Diego CA James P. Edwards - San Diego CA Sarah J. West - San Diego CA Christopher M. Tegley - San Diego CA Lin Zhi - San Diego CA Lawrence G. Hamann - San Diego CA Luc J. Farmer - La Jolla CA Robert L. Davis - Santee CA
Assignee:
Ligand Pharmaceuticals Incorporated - San Diego CA
International Classification:
A61K 3147
US Classification:
514314
Abstract:
Non-steroidal compounds which are high affinity, high selectivity modulators for steroid receptors are disclosed. Also disclosed are pharmaceutical compositions incorporating such compounds, methods for employing the disclosed compounds and compositions for treating patients requiting steroid receptor agonist or antagonist therapy, intermediates useful in the preparation of the compounds and processes for the preparation of the steroid receptor modulator compounds.
Todd K. Jones - Solana Beach CA David T. Winn - San Diego CA Lin Zhi - San Diego CA Lawrence G. Hamann - San Diego CA Christopher M. Tegley - San Diego CA Charlotte L. F. Pooley - San Diego CA
Assignee:
Ligand Pharmaceuticals Incorporated - San Diego CA
International Classification:
A61K 3147 C07D47104 C07D22116 C07D49148 C07D49152
US Classification:
514285
Abstract:
Non-steroidal compounds which are high affinity, high selectivity modulators for steroid receptors are disclosed. Also disclosed are pharmaceutical compositions incorporating such compounds, methods for employing the disclosed compounds and compositions for treating patients requiring steroid receptor agonist or antagonist therapy, intermediates useful in the preparation of the compounds and processes for the preparation of the steroid receptor modulator compounds.
Process For Preparing Steroid Receptor Modulator Compounds
Todd K. Jones - Solana Beach CA Mark E. Goldman - San Diego CA Charlotte L. F. Pooley - San Diego CA David T. Winn - San Diego CA James P. Edwards - San Diego CA Sarah J. West - San Diego CA Christopher M. Tegley - San Diego CA Lin Zhi - San Diego CA
Assignee:
Ligand Pharmaceuticals Incorporated - San Diego CA
International Classification:
C07D40104 C07D21512 C07D21518 C07D21538
US Classification:
544333
Abstract:
Non-steroidal compounds which are high affinity, high selectivity modulators for steroid receptors are disclosed. Also disclosed are pharmaceutical compositions incorporating such compounds, methods for employing the disclosed compounds and compositions for treating patients requiring steroid receptor agonist or antagonist therapy, intermediates useful in the preparation of the compounds and processes for the preparation of the steroid receptor modulator compounds.
Intermediates For Preparation Of Steroid Receptor Modulator Compounds
Todd K. Jones - Solana Beach CA David T. Winn - San Diego CA Lawrence G. Hamann - San Diego CA Lin Zhi - San Diego CA Luc J. Farmer - La Jolla CA Robert L. Davis - Santee CA
Assignee:
Ligand Pharmaceuticals Incorporated - San Diego CA
International Classification:
C07D47104
US Classification:
546 81
Abstract:
Non-steroidal compounds which are high affinity, high selectivity modulators for steroid receptors are disclosed. Also disclosed are pharmaceutical compositions incorporating such compounds, methods for employing the disclosed compounds and compositions for treating patients requiring steroid receptor agonist or antagonist therapy, intermediates useful in the preparation of the compounds and processes for the preparation of the steroid receptor modulator compounds.
Dr. Winn graduated from the Eastern Virginia Medical School Medical College in 1983. He works in Columbia, SC and specializes in Urgent Care Medicine. Dr. Winn is affiliated with Lexington Medical Center.
Dr. Winn graduated from the Northwestern University Feinberg School of Medicine in 1993. He works in San Diego, CA and specializes in Internal Medicine. Dr. Winn is affiliated with Kaiser Permanente Medical Center.