Joseph T Strupczewski

US Patent:

5602159, Feb 11, 1997

Filed:

Jun 6, 1995

Appl. No.:

8/470715

Inventors:

Edward J. Glamkowski - Warren NJ
Yulin Chiang - Covent Station NJ
Joseph T. Strupczewski - Flemington NJ
Kenneth J. Bordeau - Kintnersville PA
Peter A. Nemoto - Raritan NJ
John J. Tegeler - Bridgewater NJ

Assignee:

Hoechst-Roussel Pharmaceuticals, Inc. - Somerville NJ

International Classification:

A61K 31495
A61K 3155
A61K 31505
A61K 3144
C07D40104
C07D40300
C07D41700
C07D41900
C07D22104
C07D27504
C07D23902

US Classification:

514373

Abstract:

Heteroarylpiperidines, pyrrolidines, and piperazines are useful as antipsychotic and analgesic agents. The compounds are especially useful for treating psychoses by administering to a mammal a psychoses-treating effective amount of one of the compounds. Depot derivatives of the compounds are useful for providing long acting effects of the compounds. The compounds are also useful as analgesics by administering a pain-relieving effective amount of one of the compounds to a mammal.

US Patent:

5605913, Feb 25, 1997

Filed:

Jun 6, 1995

Appl. No.:

8/471032

Inventors:

Joseph T. Strupczewski - Flemington NJ
Yulin Chiang - Covent Station NJ
Edward J. Glamkowski - Warren NJ
Kenneth J. Bordeau - Kintnersville NJ
Grover C. Helsley - Stockton NJ

Assignee:

Hoechst Roussel Pharmaceuticals, Inc. - Somerville NJ

International Classification:

C07D40300
C07D41700
C07D41900
C07D22104
C07D40100
C07D27504
C07D23902
A61K 31495
A61K 3155
A61K 31505

US Classification:

514321

Abstract:

Heteroarylpiperidines, pyrrolidines, and piperazines are useful as antipsychotic and analgesic agents. the compounds are especially useful for treating psychoses by administering to a mammal a psychoses-treating effective amount of one of the compounds. Depot derivatives of the compounds are useful for providing long acting effects of the compounds. The compounds are also useful as analgesics by administering a pain-relieving effective amount of one of the compounds to a mammal.

US Patent:

5612342, Mar 18, 1997

Filed:

Jun 6, 1995

Appl. No.:

8/466252

Inventors:

Joseph T. Strupczewski - Flemington NJ
Kenneth J. Bordeau - Kintnersville PA

Assignee:

Hoechst-Roussel Pharmaceuticals, Inc. - Somerville NJ

International Classification:

A61K 31495
A61K 3155
A61K 31505
A61K 3144
C07D40104
C07D40304
C07D41704
C07D41904
C07D22104
C07D27504
C07D23902

US Classification:

514254

Abstract:

Heteroarylpiperidines, pyrrolidines, and piperazines are useful as antipsychotic and analgesic agents. The compounds are especially useful for treating psychoses by administering to a mammal a psychoses-treating effective amount of one of the compounds. Depot derivatives of the compounds are useful for providing long acting effects of the compounds. The compounds are also useful as analgesics by administering a pain-relieving effective amount of one of the compounds to a mammal.

US Patent:

5633265, May 27, 1997

Filed:

Jun 6, 1995

Appl. No.:

8/468993

Inventors:

Joseph T. Strupczewski - Flemington NJ
Grover C. Helsley - Stockton NJ
Edward J. Glamkowski - Warren NJ
Yulin Chiang - Covent Station NJ
Kenneth J. Bordeau - Kintnersville PA
Peter A. Nemoto - Raritan NJ
John J. Tegeler - Bridgewater NJ

Assignee:

Hoechst Marion Roussel, Inc. - Kansas City MO

International Classification:

A61K 31495
A61K 3155
A61K 31505
A61K 3144
C07D40104
C07D40304
C07D41704
C07D41904
C07D22104
C07D27504
C07D23902

US Classification:

514316

Abstract:

Heteroarylpiperidines, pyrrolidines, and piperazines are useful as antipsychotic and analgesic agents. The compounds are especially useful for treating psychoses by administering to a mammal a psychoses-treating effective amount of one of the compounds. Depot derivatives of the compounds are useful for providing long acting effects of the compounds. The compounds are also useful as analgesics by administering a pain-relieving effective amount of one of the compounds to a mammal.

US Patent:

RE37729, Jun 4, 2002

Filed:

Feb 3, 1999

Appl. No.:

09/240842

Inventors:

Edward J. Glamkowski - Warren NJ
Yulin Chiang - Convent Station NJ
Joseph T. Strupczewski - Flemington NJ
Kenneth J. Bordeau - Kintnersville PA
Peter A. Nemoto - Evanston IL
John J. Tegeler - Bridgewater NJ

Assignee:

Aventis Pharmaceuticals Inc. - Bridgewater NJ

International Classification:

A61K 31495

US Classification:

514321, 514 63, 514217, 5142338, 514249, 51425301, 51425404, 51425406, 514258, 514300, 514301, 514307, 514309, 514311, 514312, 514314, 514316, 514322, 514373, 514379, 514403, 514411, 540576, 540588, 544121, 544129, 544229, 544279, 544295, 544310, 544316, 544317, 544318, 544333, 544353, 544361, 544362, 544364, 544366, 544368, 546 14, 546 98, 546 99, 546100, 546113, 546122, 546135, 546141, 546142, 546143, 546144, 546146, 546148, 546149, 546153, 546155, 546156, 546157, 546158, 546183, 546193, 546199, 546198

Abstract:

Heteroarylpiperidines, pyrrolidines, and piperazines are useful as antipsychotic and analgesic agents. The compounds are especially useful for treating psychoses by administering to a mammal a psychoses-treating effective amount of one of the compounds. Depot derivatives of the compounds are useful for providing long acting effects of the compounds. The compounds are also useful as analgesics by administering a pain-relieving effective amount of one of the compounds to a mammal.

US Patent:

6420390, Jul 16, 2002

Filed:

Apr 19, 2000

Appl. No.:

09/556116

Inventors:

Joseph T. Strupczewski - Flemington NJ
Edward J. Glamkowski - Warren NJ
Yulin Chiang - Covent Station NJ
Kenneth J. Bordeau - Kintnersville PA
Peter A. Nemoto - Raritan NJ
John J. Tegeler - Bridgewater NJ

Assignee:

Aventis Pharmaceuticals Inc. - Bridgewater NJ

International Classification:

A61K 31445

US Classification:

514321, 514322, 546198, 546199

Abstract:

Heteroarylpiperidines, pyrrolidines, and piperazines are useful as antipsychotic and analgesic agents. the compounds are especially useful for treating psychoses by administering to a mammal a psychoses-treating effective amount of one of the compounds. Depot derivatives of the compounds are useful for providing long acting effects of the compounds. The compounds are also useful as analgesics by administering a pain-relieving effective amount of one of the compounds to a mammal.

US Patent:

RE39198, Jul 18, 2006

Filed:

Nov 15, 2000

Appl. No.:

09/712129

Inventors:

Joseph T. Strupczewski - Flemington NJ, US
Grover C. Helsley - Rosemont NJ, US
Yulin Chiang - Convent Station NJ, US
Kenneth J. Bordeau - Kintnersville PA, US
Edward J. Glamkowski - Warren NJ, US

Assignee:

Aventis Pharmaceuticals Inc. - Bridgewater NJ

International Classification:

A61K 31/445
A61K 31/495
A61K 31/42
C07D 211/00

US Classification:

514321, 51425402, 51425406, 514318, 514322, 514373, 514379, 514403, 544257, 544366, 544368, 546194, 546198, 546199, 5462701, 5462717, 548207, 5483565

Abstract:

Heteroarylpiperidines, pyrrolidines, and piperazines are useful as antipsychotic and analgesic agents. The compounds are especially useful for treating psychoses by administering to a mammal a psychoses-treating effective amounts of one of the compounds. The compounds are also useful as analgesics by administering a pain-relieving effective amount of one of the compounds to a mammal.

US Patent:

RE39265, Sep 5, 2006

Filed:

Nov 9, 2000

Appl. No.:

09/708475

Inventors:

Joseph T. Strupczewski - Flemington NJ, US
Kenneth J. Bordeau - Kintnersville PA, US
Edward J. Glamkowski - Warren NJ, US
Yulin Chiang - Convent Station NJ, US
Grover C. Helsley - Stockton NJ, US

Assignee:

Aventis Pharmaceuticals Inc. - Bridgewater NJ

International Classification:

A61P 25/04
A61K 31/495
A61K 31/55
A61K 31/44
A67K 31/505
C07D 401/04
C07D 403/04
C07D 417/04
C07D 419/04
C07D 221/04

US Classification:

51425309, 5142531, 51425404, 51425406, 514217, 5142338, 5142345, 514249, 5142581, 514269, 514274, 514296, 514300, 514301, 514307, 514309, 514311, 514312, 514314, 514321, 514322, 514373, 514379, 514403, 514411, 540576, 540588, 544121, 544129, 544132, 544135, 544137, 544279, 544295, 544316, 544317, 544318, 544333, 544353, 544361, 544362, 544364, 544366, 544367, 544368, 544371, 546 98, 546 99, 546100, 546113, 546122, 546135, 546141, 546142, 546143, 546144, 546146, 546148, 546149, 546153, 546155, 546156, 546157, 546158, 546183, 546198, 546199, 5462711, 5462721, 548110, 548207, 548209, 548219, 548221, 548241, 5483611, 5483625, 5483631

Abstract:

Heteroarylpiperidines, pyrrolidines, and piperazines are useful as antipsychotic and analgesic agents. The compounds are especially useful for treating psychoses by administering to a mammal a psychoses-treating effective amount of one of the compounds. The compounds are also useful as analgesics by administering a pain-relieving effective amount of one of the compounds to a mammal.