Manoj Nerurkar - Monmouth Junction NJ, US Vijay Naringrekar - Princeton NJ, US
Assignee:
Bristol-Myers Squibb Company - Princeton NJ
International Classification:
A61K 31/724 A61K 31/497 A61K 31/194
US Classification:
514 58, 51425407, 514574
Abstract:
An aripiprazole formulation is provided which includes the antipsychotic agent aripiprazole in the form of an inclusion complex in a β-cyclodextrin, preferably, sulfobutyl ether β-cyclodextrin (SBECD), which in the form of an injectable produces reversible generally minimal to mild irritation at the intramuscular injection site. A method for minimizing or reducing irritation caused by aripiprazole at an intramuscular injection site and a method for treating schizophrenia employing the above formulation are also provided.
Controlled Release Sterile Injectable Aripiprazole Formulation And Method
Janusz W. Kostanski - Princeton NJ, US Takakuni Matsuda - Tokushima, JP Manoj Nerurkar - Monmouth Junction NJ, US Vijay H. Naringrekar - Princeton NJ, US
Assignee:
Otsuka Pharmaceutical Co., Ltd. - Tokyo
International Classification:
A61K 31/497
US Classification:
51425307, 51425303, 5142521
Abstract:
A controlled release sterile freeze-dried aripiprazole formulation is provided which is formed of aripiprazole of a desired mean particle size and a vehicle therefor, which upon constitution with water and intramuscular injection releases aripiprazole over a period of at least about one week and up to about eight weeks. A method for preparing the controlled release freeze-dried aripiprazole formulation, and a method for treating schizophrenia employing the above formulation are also provided.
Controlled Release Sterile Injectable Aripiprazole Formulation And Method
Janusz W. Kostanski - Princeton NJ, US Takakuni Matsuda - Tokushima, JP Manoj Nerurkar - Monmouth Junction NJ, US Vijay H. Naringrekar - Princeton NJ, US
Assignee:
Otsuka Pharmaceutical Co., Ltd. - Tokyo
International Classification:
A61K 31/497
US Classification:
51425307, 51425303, 5142521
Abstract:
A controlled release sterile freeze-dried aripiprazole formulation is provided which is formed of aripiprazole of a desired mean particle size and a vehicle therefor, which upon constitution with water and intramuscular injection releases aripiprazole over a period of at least about one week and up to about eight weeks. A method for preparing the controlled release freeze-dried aripiprazole formulation, and a method for treating schizophrenia employing the above formulation are also provided.
Controlled Release Sterile Injectable Aripiprazole Formulation And Method
Janusz W. Kostanski - Princeton NJ, US Takakuni Matsuda - Tokushima, JP Manoj Nerurkar - Monmouth Junction NJ, US Vijay H. Naringrekar - Princeton NJ, US
Assignee:
Otsuka Pharmaceutical Co., Ltd. - Tokyo
International Classification:
A61K 31/497
US Classification:
51425307, 51425303, 5142521
Abstract:
A controlled release sterile freeze-dried aripiprazole formulation is provided which is formed of aripiprazole of a desired mean particle size and a vehicle therefor, which upon constitution with water and intramuscular injection releases aripiprazole over a period of at least about one week and up to about eight weeks. A method for preparing the controlled release freeze-dried aripiprazole formulation, and a method for treating schizophrenia employing the above formulation are also provided.
Manoj Nerurkar - Monmouth Junction NJ, US Vijay Naringrekar - Paramus NJ, US Mark Dominick - Evansville IN, US
International Classification:
A61K031/724 C08B037/16
US Classification:
514/058000, 536/046000
Abstract:
An aripiprazole formulation is provided which includes the antipsychotic agent aripiprazole in the form of an inclusion complex in a -cyclodextrin, preferably, sulfobutyl ether -cyclodextrin (SBECD), which in the form of an injectable produces reversible generally minimal to mild irritation at the intramuscular injection site. A method for minimizing or reducing irritation caused by aripiprazole at an intramuscular injection site and a method for treating schizophrenia employing the above formulation are also provided.
Controlled Release Sterile Injectable Aripiprazole Formulation And Method
Janusz Kostanski - Princeton NJ, US Takakuni Matsuda - Tokushima, JP Manoj Nerurkar - Monmouth Junction NJ, US Vijay Naringrekar - Princeton NJ, US
International Classification:
A61K 31/496 A61K 9/00
US Classification:
424400000, 514253070
Abstract:
A controlled release sterile freeze-dried aripiprazole formulation is provided which is formed of aripiprazole of a desired mean particle size and a vehicle therefor, which upon constitution with water and intramuscular injection releases aripiprazole over a period of at least about one week and up to about eight weeks. A method for preparing the controlled release freeze-dried aripiprazole formulation, and a method for treating schizophrenia employing the above formulation are also provided.
Manoj NERURKAR - Monmouth Junction NJ, US Vijay NARINGREKAR - Princeton NJ, US
International Classification:
A61K 31/497 A61P 43/00
US Classification:
51425308
Abstract:
An aripiprazole formulation is provided which includes the antipsychotic agent aripiprazole in the form of an inclusion complex in a β-cyclodextrin, preferably, sulfobutyl ether β-cyclodextrin (SBECD), which in the form of an injectable produces reversible generally minimal to mild irritation at the intramuscular injection site. A method for minimizing or reducing irritation caused by aripiprazole at an intramuscular injection site and a method for treating schizophrenia employing the above formulation are also provided.
Controlled Release Sterile Injectable Aripiprazole Formulation And Method
Janusz W. Kostanski - Princeton NJ, US Takakuni Matsuda - Tokushima, JP Manoj Nerurkar - Monmouth Junction NJ, US Vijay H. Naringrekar - Princeton NJ, US
Assignee:
OTSUKA PHARMACEUTICAL CO., LTD. - Tokyo
International Classification:
A61K 31/496 A61P 25/18 A61K 9/14
US Classification:
424400, 51425307
Abstract:
A controlled release sterile freeze-dried aripiprazole formulation is provided which is formed of aripiprazole of a desired mean particle size and a vehicle therefor, which upon constitution with water and intramuscular injection releases aripiprazole over a period of at least about one week and up to about eight weeks. A method for preparing the controlled release freeze-dried aripiprazole formulation, and a method for treating schizophrenia employing the above formulation are also provided.